Bioactive Small Molecules for Ion Channels, GPCRs & Transporters

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Bioactive Small Molecules for Ion Channels, GPCRs & Transporters

Search by Target or keyword to jump directly into the full catalog results, scoped to Alomone Labs.

Featured Small Molecules

11 featured items

Nav Tetrodotoxin citrate
TTX-100
Tetrodotoxin citrate
Nav blocker
From$430
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TRPV1 Capsaicin
CAP-TRPV1
Capsaicin
TRPV1 agonist
From$626
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AMPA/Kainate CNQX disodium salt
CNQX-Na
CNQX disodium salt
AMPA/Kainate antagonist
From$40
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AMPA DNQX
DNQX
DNQX
AMPA antagonist
From$37
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AMPA/Kainate NBQX disodium salt
NBQX-Na
NBQX disodium salt
AMPA/Kainate antagonist
From$37
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TRPA1 HC-030031
HC-030031
HC-030031
TRPA1 antagonist
From$50
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TRPV1 SB-366791
SB-366791
SB-366791
TRPV1 antagonist
From$85
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KCNQ XE991 dihydrochloride
XE991-2HCl
XE991 dihydrochloride
KCNQ blocker
From$132
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Nav Veratridine
VERA
Veratridine
Nav activator
From$103
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KCa3.1 TRAM 34
TRAM34
TRAM 34
KCa3.1 inhibitor
From$110
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ET-B BQ788 sodium salt
BQ788-Na
BQ788 sodium salt
Endothelin ET-B antagonist
From$134
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Popular Targets

  • TRP channel ligands (TRPV1 / TRPA1 / TRPM8)
  • Voltage-gated sodium channel modulators (Nav)
  • AMPA / NMDA receptor agents
  • Calcium channel blockers (L-type, T-type)

What's Included

  • Certificate of Analysis
  • Stability & storage guidance
  • Peer-reviewed references
  • Cold-chain shipping options

Small Molecules: FAQ

Match the mechanism to your assay question. Use an agonist when you want to activate the target channel or receptor to study its downstream effects, and an antagonist when you need to block or inhibit the target to observe loss-of-function outcomes.
Each product datasheet includes recommended solvents, stock solution concentrations, and working concentrations. Most compounds are available as lyophilized powder; some are offered pre-dissolved for convenience.
Protect from light and moisture, store desiccated at the temperature indicated on the datasheet (typically −20 °C). Aliquot stock solutions upon first reconstitution to avoid repeated freeze–thaw cycles.