| Field | Specification |
|---|---|
| Mfr No | |
| Activity | |
| Alternative Names | TD-1211 |
| Cas No. | |
| Molecular Weight | |
| Product Type | |
| Signaling Pathway | |
| SMILES | |
| Target |
Compound Overview
Axelopran (CAS 949904-48-7) is a research-grade small molecule supplied by TargetMol.
Alternative names: TD-1211
Physical Properties
| CAS Number | 949904-48-7 |
|---|---|
| Molecular Formula | C26H39N3O4 |
| Molecular Weight | 457.61 g/mol |
| SMILES | C(CN(CC1CCCCC1)C((CH)(CO)O)=O)N2(C)3(C(CH)(C(C)2(CC3)(H))C4=CC(C(N)=O)… |
| Form | Solid |
| Shipping | Room Temperature (RT) |
Biological Activity
Axelopran(TD-1211) is potentially useful for the treatment of opioid-induced constipation, it is a potent, selective, and peripherally-restricted u-, kappa-, and delta-opioid receptor antagonist.
Safety & Regulatory
For Research Use Only (RUO). Not for therapeutic, diagnostic, or clinical use. Wear appropriate PPE and consult the Safety Data Sheet (SDS) prior to handling.
It is recommended to sonicate at a lower frequency
For currently available products, batch-specific purity data (HPLC chromatogram, NMR spectrum, and Certificate of Analysis) is accessible via the DataSheet link on the product page. For future or custom synthesis products, purity determination is conducted upon availability and published on the product page. Contact BioHippo for batch-specific CoA requests or custom synthesis enquiries.
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- Add-on labels & handles: D/¹³C/¹⁵N isotopes (LC-MS/internal standards), azide/alkyne or other functional handles for conjugation
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