Rimonabant

SKU:BHB11900309
Suppliers
StressMarq Biosciences Inc.
StressMarq Biosciences Inc.
Details Products
Overview
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Rimonabant is a research-grade small-molecule inhibitor of CB1 Receptor supporting Cell signaling and Neuroscience research. Supplied as a white powder with >98% purity (CAS 158681-13-1, MW 463.8) soluble in DMSO; store at -20°C. For research use only.
Cas No. 158681-13-1
Molecular Formula C22H21Cl3N4O
Purity >98% (TLC); NMR (Conforms)
Application Notes CB1 Receptor Antagonist
Options selector
Catalog no. Size
SIH-528-5MG 5 mg
SIH-528-25MG 25 mg
Available Options

Select the variant that best fits your experiment. Availability and lead time may vary by option.

  • Options: Size (2) — 25 mg, 5 mg.
  • Lead time: options listed as “in stock at manufacturer” typically ship in 2-3 business days; other statuses may take longer.
  • Storage: -20ºC
  • Shipping: ships at ambient temperature.
  • Upon receipt: store at the recommended temperature as soon as possible.
  • Sales terms and conditions: Please review prior to ordering.
Field Specification
Mfr No SIH-528
Activity
  • Inhibitor
Alternative Names 5-(4-Chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-N-1-piperidinyl-1H-pyrazole-3-carboxamide hydrochloride, SR-141716, SR-141716A, SR141716, SR141716A
Cas No. 158681-13-1
Form White powder
Molecular Weight 463.8
Product Type
  • Biochemicals
  • Small Molecules
Purity >98% (TLC); NMR (Conforms)
Shipping Shipped Ambient
SMILES Cc1c(n(nc1C(=O)NN2CCCCC2)c3ccc(cc3Cl)Cl)c4ccc(cc4)Cl
Solubility Soluble in DMSO (50 mg/ml)
Source Synthetic
Storage -20ºC

Rimonabant is a selective cannabinoid receptor type 1 (CB1) antagonist that was originally developed as an anti-obesity drug. In neuroscience, it has been studied for its effects on the endocannabinoid system, which plays a critical role in mood regulation, appetite, and neuroprotection. Rimonabant's ability to modulate CB1 receptor signaling has implications for treating neuropsychiatric disorders, including depression and anxiety. Additionally, its influence on neuroinflammation and synaptic plasticity positions it as a candidate for research in neurodegenerative diseases, although its clinical use has been limited due to psychiatric side effects.

Details:

Classification

D1B Toxic Material Causing Immediate and Serious Toxic Effects - Toxic by ingestion

D2B Toxic Material Causing Other Toxic Effects - Moderate eye irritant

Hazard statement(s):

  • H301 Toxic if swallowed.
  • H319 Causes serious eye irritation.

Precautionary statement(s):

  • P301 + P310 IF SWALLOWED: Immediately call a POISON CENTER or doctor/ physician.
  • P305 + P351 + P338 IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continue rinsing.

Rimonabant (StressMarq Biosciences Inc., Victoria BC CANADA, Catalog # SIH-528)

Need this compound in a format that drops straight into your assay? We can tailor formulation, chemistry, and documentation so your results stay consistent across runs and re-orders.

  • Format options: solid or pre-dissolved solution (choose solvent), target concentration, aliquots, light/moisture-protected packaging
  • Chemistry options: free base/acid vs salt forms, hydrate/solvate preference, stereoisomer control (single enantiomer or racemate), close analogs
  • Add-on labels & handles: D/¹³C/¹⁵N isotopes (LC-MS/internal standards), azide/alkyne or other functional handles for conjugation
  • QC & documentation: standard COA or enhanced analytical pack (HPLC/LC-MS/NMR), chiral purity, residual solvents, water content (KF), method-specific specs
  • Scale & continuity: mg to gram scale, bulk pricing, lot reservation, repeat-order continuity

To quote quickly, tell us: compound name + CAS/structure (SMILES or mol file), intended assay context, solvent preference, salt/stereochemistry requirements, purity/QC level, and the amount (mg–g).

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