| Field | Specification |
|---|---|
| Mfr No | |
| Activity | |
| Alternative Names | HSK3486 |
| Cas No. | |
| Molecular Weight | |
| Product Type | |
| Signaling Pathway | |
| SMILES | |
| Target |
Compound Overview
Cipepofol (CAS 1637741-58-2) is a research-grade small molecule supplied by TargetMol.
Alternative names: HSK3486
Physical Properties
| CAS Number | 1637741-58-2 |
|---|---|
| Molecular Formula | C14H20O |
| Molecular Weight | 204.31 g/mol |
| SMILES | (CH)(C)(C1=C(O)C(C(C)C)=CC=C1)C2CC2 |
| Form | Solid |
| Shipping | Room Temperature (RT) |
Biological Activity
Cipepofol (HSK3486) is a GABAA receptor agonist with sedative properties and protective effects in a variety of cardiovascular diseases.Cipepofol activates the Sirtuin1 (Sirt1)/Nrf2 pathway and induces apoptosis in cardiomyocytes, and can be used to study myocardial infarction, myocardial ischemia/reperfusion injury, and octopus pot syndrome.
Target(s): Apoptosis, GABA Receptor
Signaling pathway(s): Apoptosis, Membrane transporter/Ion channel, Neuroscience
Safety & Regulatory
For Research Use Only (RUO). Not for therapeutic, diagnostic, or clinical use. Wear appropriate PPE and consult the Safety Data Sheet (SDS) prior to handling.
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