| Field | Specification |
|---|---|
| Target | |
| CAS no. | |
| Applications | |
| Molecular weight | |
| Molecular formula | C27H32ClNO4 |
| Purity | |
| SMILES | |
| Form | Liquid |
| Storage | |
| Shipping | |
| Catalog no. (Mfr.) | |
| Main SKU |
Compound Overview
EP4 receptor agonist 2 is a potent EP4 receptor agonist with an EC50 of 0.8 nM and Ki values of >100000 nM, 38000 nM and 3.1 nM at EP2, EP3 and EP4, respectively[1]. It is supplied as a colorless to light yellow liquid (C27H32ClNO4, MW 470.00) at 99.0% purity.
Physical & Chemical Properties
| CAS Number | 493035-81-7 |
|---|---|
| Molecular Formula | C27H32ClNO4 |
| Molecular Weight | 470.00 g/mol |
| Purity | 99.0% |
| Appearance | Liquid |
| Color | Colorless to light yellow |
| SMILES | CC1=C(C=CC(Cl)=C1)C2=CC(C(O)/C=C/[C@@H]3N(C(CC3)=O)CCCCCCC(O)=O)=CC=C2 |
| Target | EP4, EP2, EP3 |
| Signaling Pathway | GPCR/G Protein |
| Storage | Solution, -20°C, 2 years. |
| Shipping | Room temperature in continental US; may vary elsewhere. |
Biological Activity
IC50 & Target[1]
|
EP4 0.8 nM (EC50) |
EP2 >100000 nM (Ki) |
EP3 38000 nM (Ki) |
EP4 3.1 nM (Ki) |
Literature Cited
Sources cited in this description. Peer-reviewed publications that used this product are listed under References.
Safety
For Research Use Only. Not for use in diagnostic or therapeutic procedures, and not for human or veterinary use. Handle in accordance with the Safety Data Sheet and your institution's chemical hygiene plan.
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