| Field | Specification |
|---|---|
| CAS no. | |
| Applications | |
| Molecular weight | |
| Molecular formula | C18H17N3 |
| SMILES | |
| Storage | |
| Shipping | |
| Catalog no. (Mfr.) | |
| Main SKU |
Compound Overview
FR252384 is a neuropeptide Y-Y5 receptor antagonist, with an IC50 of 2.3 nM. Its molecular formula is C18H17N3, with a molecular weight of 275.35 g/mol.
Physical & Chemical Properties
| CAS Number | 447405-11-0 |
|---|---|
| Molecular Formula | C18H17N3 |
| Molecular Weight | 275.35 g/mol |
| SMILES | CC1=CC=C(CCC2)C(C3=C2N=C(C4=CC=CN=C4)N3)=C1 |
| Signaling Pathway | GPCR/G Protein; Neuronal Signaling |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Shipping | Room temperature in continental US; may vary elsewhere. |
Biological Activity
IC50 & Target
IC50: 2.3 nM (neuropeptide Y-Y5 receptor)[1]
Literature Cited
Sources cited in this description and in the In Vitro & In Vivo Data tab. Peer-reviewed publications that used this product are listed under References.
Safety
For Research Use Only. Not for use in diagnostic or therapeutic procedures, and not for human or veterinary use. Handle in accordance with your institution's chemical hygiene plan.
In Vivo
FR252384 is absorbed orally and can cross into the brain[1].
Data provided by the manufacturer. Numbered citations refer to the Literature Cited list in the product description.
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