| Field | Specification |
|---|---|
| Applications | |
| Molecular weight | |
| Molecular formula | C21H23N3O |
| SMILES | |
| Storage | |
| Shipping | |
| Catalog no. (Mfr.) | |
| Main SKU |
Compound Overview
HIF-1α-IN-6 is an inhibitor of HIF-1α, with IC50 values of 0.6 nM and 53.3 nM in MiaPaCa-2 and MDA-MB-231 cells, respectively. It can reduce HIF-1α expression by decreasing HIF-1α mRNA levels[1]. It has a molecular formula of C21H23N3O and a molecular weight of 333.43 g/mol.
Physical & Chemical Properties
| Molecular Formula | C21H23N3O |
|---|---|
| Molecular Weight | 333.43 g/mol |
| SMILES | CC1=NC2=CC(OC)=CC=C2C(NC3=CC=CC(N4CCCC4)=C3)=C1 |
| Signaling Pathway | Metabolic Enzyme/Protease |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
| Shipping | Room temperature in continental US; may vary elsewhere. |
Literature Cited
Sources cited in this description. Peer-reviewed publications that used this product are listed under References.
Safety
For Research Use Only. Not for use in diagnostic or therapeutic procedures, and not for human or veterinary use. Handle in accordance with your institution's chemical hygiene plan.
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