Promethazine

SKU:BHB20400395
Overview
Click light‑blue chips for details
Promethazine (CAS 60-87-7) is a receptor modulator supplied as a solid powder by TargetMol. For biochemical profiling and cell-based assay applications.
Activity Receptor Modulator
CAS No. 60-87-7
Molecular Weight 284.42 g/mol
Form Solid
Shipping Room Temperature
Options selector
Catalog no. Size
T0445-5MG 5 mg
T0445-1MLX10MM 1 mL x 10 mM (in DMSO)
T0445-10MG 10 mg
T0445-25MG 25 mg
T0445-50MG 50 mg
T0445-100MG 100 mg
T0445-500MG 500 mg
Available Options

Select the variant that best fits your experiment. Availability and lead time may vary by option.

  • Options: Size: 5 mg, 1 mL x 10 mM (in DMSO), 10 mg, 25 mg, 50 mg, 100 mg, 500 mg
  • Lead time: In Stock at Manufacturer — options listed in "Availability Content"; other statuses may take longer.
  • Storage: −20 °C
  • Shipping: Room temperature (RT) shipment.
  • Upon receipt: Store at −20 °C as soon as possible.
  • Sales terms and conditions: Please review prior to ordering.
Field Specification
Mfr No T0445
Activity
  • Receptor Modulator
Alternative Names Proazamine
Cas No. 60-87-7
Molecular Weight 284.42
Product Type
  • Small Molecule Inhibitor
Signaling Pathway GPCR/G Protein///Immunology/Inflammation///Neuroscience
SMILES C(C(N(C)C)C)N1C=2C(SC=3C1=CC=CC3)=CC=CC2
Target Histamine Receptor///Adrenergic Receptor///AChR///CaMK///Dopamine Receptor///5-HT Receptor

Compound Overview

Promethazine (CAS 60-87-7) is a research-grade small molecule supplied by TargetMol.

Alternative names: Proazamine

Physical Properties

CAS Number 60-87-7
Molecular Formula C17H20N2S
Molecular Weight 284.42 g/mol
SMILES C(C(N(C)C)C)N1C=2C(SC=3C1=CC=CC3)=CC=CC2
Form Solid
Shipping Room Temperature (RT)

Biological Activity

Promethazine (Proazamine) is an analogue of anti-glaucoma prostaglandin (PG) .

Target(s): Histamine Receptor, Adrenergic Receptor, AChR, CaMK, Dopamine Receptor, 5-HT Receptor

Signaling pathway(s): GPCR/G Protein, Immunology/Inflammation, Neuroscience

Safety & Regulatory

For Research Use Only (RUO). Not for therapeutic, diagnostic, or clinical use. Wear appropriate PPE and consult the Safety Data Sheet (SDS) prior to handling.

Can inhibitors be used for cell experiments?

Yes — TargetMol inhibitors can be used in cell-based and in vitro experiments. Prepare a DMSO stock, then dilute into cell culture medium to the desired working concentration, keeping DMSO ≤ 0.1% (v/v) to avoid solvent toxicity. Note that not all compounds have published data for every cell line or assay system; in such cases, perform a dose-response experiment with appropriate positive and vehicle controls to validate efficacy in your specific model.

Can inhibitors be used for animal experiments?

Yes, our inhibitors can be used for animal/in vivo experiments. However, some compounds may not have literature supporting their use in animal experiments. In such cases, we cannot guarantee efficacy.

Need this compound in a format that drops straight into your assay? We can tailor formulation, chemistry, and documentation so your results stay consistent across runs and re-orders.

  • Format options: solid or pre-dissolved solution (choose solvent), target concentration, aliquots, light/moisture-protected packaging
  • Chemistry options: free base/acid vs salt forms, hydrate/solvate preference, stereoisomer control (single enantiomer or racemate), close analogs
  • Add-on labels & handles: D/¹³C/¹⁵N isotopes (LC-MS/internal standards), azide/alkyne or other functional handles for conjugation
  • QC & documentation: standard COA or enhanced analytical pack (HPLC/LC-MS/NMR), chiral purity, residual solvents, water content (KF), method-specific specs
  • Scale & continuity: mg to gram scale, bulk pricing, lot reservation, repeat-order continuity

To quote quickly, tell us: compound name + CAS/structure (SMILES or mol file), intended assay context, solvent preference, salt/stereochemistry requirements, purity/QC level, and the amount (mg–g).

Can’t find the compound you’re looking for?
Send the CAS or structure and your specs. We can help source it, suggest close equivalents, or discuss custom synthesis with the right QC documentation (RUO).

Get a Quote

Please use this form for bulk quantity requests or customized products.

Contact Information

Product Information

Try Celltrypse Free – Request Your Sample Today

Experience the power of Celltrypse™, c-LEcta's innovative enzyme solution for gentle and efficient cell dissociation. Request your free sample and discover a superior alternative for your cell culture workflows.

Try Celltrypse Free – Request Your Sample Today

Try Celltrypse Free – Request Your Sample Today

Experience the power of Celltrypse™, c-LEcta's innovative enzyme solution for gentle and efficient cell dissociation. Request your free sample and discover a superior alternative for your cell culture workflows.

Try Celltrypse Free – Request Your Sample Today