SC-53116

SKU:BHB21900588
Overview
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SC-53116 (CAS 141196-99-8) is an agonist. Reported to act on 5-HT 4 Receptor. Relevant to GPCR/G Protein and Neuronal Signaling research. Molecular formula C16H22ClN3O2, molecular weight 323.82 g/mol.
CAS Number 141196-99-8
Molecular Weight 323.82 g/mol
Target 5-HT 4 Receptor
Storage See Certificate of Analysis
Options selector
Catalog no. Size
HY-123747-50MG 50 mg
HY-123747-100MG 100 mg
HY-123747-250MG 250 mg
Available Options

Select the variant that best fits your experiment. Availability and lead time may vary by option.

  • Options: Size: 50 mg, 100 mg, 250 mg
  • Lead time: confirmed on inquiry for every option.
  • Storage: Please store the product under the recommended conditions in the Certificate of Analysis.
  • Shipping: Room temperature in continental US; may vary elsewhere.
  • Upon receipt: store as stated on the Certificate of Analysis; contact us if you need the condition before ordering.
Field Specification
Target 5-HT 4 Receptor
CAS no. 141196-99-8
Applications
  • Functional Assay (In Vitro)
Molecular weight 323.82
Molecular formula C16H22ClN3O2
SMILES O=C(C1=CC(Cl)=C(C=C1OC)N)NC[C@H]2[C@@]3(CCCN3CC2)[H]
Storage Refer to Certificate of Analysis (CoA) for storage conditions
Shipping Room temperature in continental US; may vary elsewhere.
Catalog no. (Mfr.) HY-123747
Main SKU BHB21900588
Agonists

Compound Overview

SC-53116 is a selective 5-HT4 receptor agonist, with an EC50 of 23 nM[1]. It has the molecular formula C16H22ClN3O2 and a molecular weight of 323.82 g/mol.

Physical & Chemical Properties

CAS Number 141196-99-8
Molecular Formula C16H22ClN3O2
Molecular Weight 323.82 g/mol
SMILES O=C(C1=CC(Cl)=C(C=C1OC)N)NC[C@H]2[C@@]3(CCCN3CC2)[H]
Target 5-HT 4 Receptor
Signaling Pathway GPCR/G Protein; Neuronal Signaling
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
Shipping Room temperature in continental US; may vary elsewhere.

Biological Activity

Activity & Target

5-HT4 Receptor

23 nM (EC50)

Literature Cited

Sources cited in this description. Peer-reviewed publications that used this product are listed under References.

[1]. Becker DP, et al. Bridgehead-methyl analog of SC-53116 as a 5-HT4 agonist. Bioorg Med Chem Lett. 2004 Jun 21;14(12):3073-5.

Safety

For Research Use Only. Not for use in diagnostic or therapeutic procedures, and not for human or veterinary use. Handle in accordance with your institution's chemical hygiene plan.

Q.Why is there no price listed?
A.Every size of this product is quoted on inquiry. Send us the size you need and we will come back with price and lead time.
Q.Can this be used in humans or for diagnostics?
A.No. This product is supplied For Research Use Only. It is not for diagnostic or therapeutic procedures and not for human or veterinary use.

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