Oncology Signaling — Biochemicals

310Products
310 products
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Cbz-B3A – Figure 1 of 1
Target: mTOR
Small Molecule Inhibitor Functional Assay (In Vitro)
From $108.00
Regular price From $108.00
In Stock at Manufacturer
BRD7389 – Figure 1 of 1
Target: DAPK///S6 Kinase///Pim///FLT///SGK///CDK
Small Molecule Inhibitor Functional Assay (In Vitro)
From $29.00
Regular price From $29.00
In Stock at Manufacturer
Sitravatinib malate – Figure 1 of 1
Target: TAM Receptor
Small Molecule Inhibitor Functional Assay (In Vitro)
From $1,520.00
Regular price From $1,520.00
Made to order
Cromolyn sodium – Figure 1 of 1
Target: GSK-3///Potassium Channel///Calcium Channel///Others
Small Molecule Inhibitor Functional Assay (In Vitro)
$48.00
Regular price $48.00
In Stock at Manufacturer
PI3K-IN-10 – Figure 1 of 1
Target: PI3K
Small Molecule Inhibitor Functional Assay (In Vitro)
Made to order
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JTV-519 hemifumarate – Figure 1 of 1
Target: MELK
Small Molecule Inhibitor Functional Assay (In Vitro)
Made to order
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bpV(phen) – Figure 1 of 1
Target: PTEN
Small Molecule Inhibitor Functional Assay (In Vitro)
$1,520.00
Regular price $1,520.00
Made to order
CK2/ERK8-IN-1 – Figure 1 of 1
Target: DYRK///Casein Kinase///Pim///Apoptosis///ERK
Small Molecule Inhibitor Functional Assay (In Vitro)
From $0.00
Regular price From $0.00
In Stock at Manufacturer
c-Fms-IN-8 – Figure 1 of 1
Target: CSF-1R
Small Molecule Inhibitor Functional Assay (In Vitro)
From $1,400.00
Regular price From $1,400.00
Made to order
Kanosamine hydrochloride – Figure 1 of 1
Target: Akt
Small Molecule Inhibitor Functional Assay (In Vitro)
From $98.00
Regular price From $98.00
Made to order
Gartisertib – Figure 1 of 1
Target: ATM/ATR
Small Molecule Inhibitor Functional Assay (In Vitro)
From $129.00
Regular price From $129.00
In Stock at Manufacturer
LY-2584702 hydrochloride – Figure 1 of 1
Target: S6 Kinase
Small Molecule Inhibitor Functional Assay (In Vitro)
From $1,520.00
Regular price From $1,520.00
Made to order
Charantin – Figure 1 of 1
Target: GSK-3
Small Molecule Inhibitor Functional Assay (In Vitro)
Discontinued
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Trichostatin A – Figure 1 of 2
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $129.00
Regular price From $129.00
In Stock at Manufacturer
Thapsigargin Epoxide – Figure 1 of 1
Target: SERCA pump
Biochemicals, Small Molecules Functional Assay (In Vitro)
$261.00
Regular price $261.00
In Stock at Manufacturer
PMA – Figure 1 of 2
PMA
Target: Protein kinase C
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $103.00
Regular price From $103.00
In Stock at Manufacturer
NS-1619 – Figure 1 of 2
Target: KCa1.1 channel, SERCA pump
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $91.00
Regular price From $91.00
In Stock at Manufacturer
Geldanamycin – Figure 1 of 2
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $120.00
Regular price From $120.00
In Stock at Manufacturer
Gambogic acid – Figure 1 of 2
Target: Caspase, Bcl-2, Bax, CD71, Kir2.1 channel
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $66.00
Regular price From $66.00
In Stock at Manufacturer
Gambogic amide – Figure 1 of 2
Target: TrkA receptor
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $117.00
Regular price From $117.00
In Stock at Manufacturer
A-740003 – Figure 1 of 2
Target: P2X7 receptor
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $50.00
Regular price From $50.00
In Stock at Manufacturer
17-AAG – Figure 1 of 2
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $188.00
Regular price From $188.00
In Stock at Manufacturer
Arvanil – Figure 1 of 2
Target: TRPV1 channel, CB1 receptor
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $50.00
Regular price From $50.00
In Stock at Manufacturer
D-3263 hydrochloride – Figure 1 of 2
Target: TRPM8 channel
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $235.00
Regular price From $235.00
In Stock at Manufacturer
Chemical structure of Duloxetine HCl (SIH-549), a 5-HT-noradrenaline reuptake inhibitor. CAS #: 136434-34-9. Molecular Formula: C18H19NOS.HCl. Molecular Weight: 333.9 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $57.00
Regular price From $57.00
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Chemical structure of Stattic (SIH-554), a STAT3 inhibitor. CAS #: 19983-44-9. Molecular Formula: C8H5NO4S. Molecular Weight: 211.2 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $57.00
Regular price From $57.00
In Stock at Manufacturer
Chemical structure of BSI 201 (SIH-539), a PARP1 inhibitor. CAS #: 160003-66-7. Molecular Formula: C7H5IN2O3. Molecular Weight: 292 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $80.00
Regular price From $80.00
In Stock at Manufacturer
Chemical structure of Pazopanib (SIH-506), a Multi target receptor tyrosine kinase inhibitor. CAS #: 44473-52-6. Molecular Formula: C21H23N7O2S. Molecular Weight: 437.5 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $87.00
Regular price From $87.00
In Stock at Manufacturer
Chemical structure of LY364947 (SIH-504), a ALK5 kinase inhibitor. CAS #: 396129-53-6. Molecular Formula: C17H12N4. Molecular Weight: 272.3 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $92.00
Regular price From $92.00
In Stock at Manufacturer
Chemical structure of Pepstatin A (SIH-533), a Aspartic protease inhibitor. CAS #: 26305-03-3. Molecular Formula: C34H63N5O9. Molecular Weight: 685.9 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $68.00
Regular price From $68.00
In Stock at Manufacturer
Chemical structure of Leptomycin B (SIH-534), a Nuclear export inhibitor. CAS #: 87081-35-4. Molecular Formula: C33H48O6. Molecular Weight: 540.7 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $87.00
Regular price From $87.00
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Chemical structure of Bexarotene (SIH-535), a Retinoid RXR agonist. CAS #: 153559-49-0. Molecular Formula: C24H28O2. Molecular Weight: 348.5 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $74.00
Regular price From $74.00
In Stock at Manufacturer
Chemical structure of LH 846 (SIH-503), a Casein kinase 1d inhibitor. CAS #: 639052-78-1. Molecular Formula: C16H13ClN2OS. Molecular Weight: 316.8 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $79.00
Regular price From $79.00
In Stock at Manufacturer
Chemical structure of ZM 306416 (SIH-487), a VEGFR kinase inhibitor. CAS #: 690206-97-4. Molecular Formula: C16H13ClFN3O2. Molecular Weight: 333.7 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $87.00
Regular price From $87.00
In Stock at Manufacturer
Chemical structure of WY-14643 (SIH-531), a PPAR alpha agonist. CAS #: 50892-23-4. Molecular Formula: C14H14ClN3O2S. Molecular Weight: 323.8 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $98.00
Regular price From $98.00
In Stock at Manufacturer
Chemical structure of Terazosin Hydrochloride (SIH-516), a Alpha adrenergic antagonist, and Hsp90 Activator. CAS #: 63074-08-8. Molecular Formula: C19H25N5O4 · HCl. Molecular Weight: 423.89 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $63.00
Regular price From $63.00
In Stock at Manufacturer

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