Cardiovascular Biochemicals

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50 products
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Tyrphostin AG 1296 – Figure 1 of 2
Target: PDGFR receptor
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $75.00
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SB209670 – Figure 1 of 2
Target: Endothelin receptor
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $235.00
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IRL 2500 – Figure 1 of 2
Target: ET-B receptor
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $134.00
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A-803467 – Figure 1 of 2
Target: NaV1.8 channel
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $66.00
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Darusentan – Figure 1 of 2
Target: ET-A receptor
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $235.00
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BQ-123 trifluoroacetate – Figure 1 of 2
Target: ET-A receptor
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $235.00
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BQ-123 sodium salt – Figure 1 of 2
Target: ET-A receptor
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $168.00
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Chemical structure of Duloxetine HCl (SIH-549), a 5-HT-noradrenaline reuptake inhibitor. CAS #: 136434-34-9. Molecular Formula: C18H19NOS.HCl. Molecular Weight: 333.9 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of ML297 (SIH-553), a GIRK activator. CAS #: 1443246-62-5. Molecular Formula: C17H14F2N4O. Molecular Weight: 328.32 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of LY364947 (SIH-504), a ALK5 kinase inhibitor. CAS #: 396129-53-6. Molecular Formula: C17H12N4. Molecular Weight: 272.3 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of Bexarotene (SIH-535), a Retinoid RXR agonist. CAS #: 153559-49-0. Molecular Formula: C24H28O2. Molecular Weight: 348.5 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of ZM 306416 (SIH-487), a VEGFR kinase inhibitor. CAS #: 690206-97-4. Molecular Formula: C16H13ClFN3O2. Molecular Weight: 333.7 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of SU1498 (SIH-480), a VEGFR kinase inhibitor. CAS #: 168835-82-3. Molecular Formula: C25H30N2O2. Molecular Weight: 390.5 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of Vatalanib Dihydrochloride (SIH-484), a VEGFRK inhibitor. CAS #: 212141-51-0. Molecular Formula: C20H17Cl3N4. Molecular Weight: 419.7 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $74.00
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Chemical structure of ML167 (SIH-505), a Clk4 kinase inhibitor. CAS #: 1285702-20-6. Molecular Formula: C19H17N3O3. Molecular Weight: 335.4 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of Ruxolitinib (SIH-509), a JAK kinase inhibitor. CAS #: 941678-49-5. Molecular Formula: C17H18N6. Molecular Weight: 306.4 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of PD325901 (SIH-507), a MEK kinase inhibitor. CAS #: 391210-10-9. Molecular Formula: C16H14F3IN2O4. Molecular Weight: 482.2 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of SU 4312 (SIH-481), a VEGFR / PDGFR kinase inhibitor. CAS #: 5812-07-7. Molecular Formula: C17H16N2O. Molecular Weight: 264.3 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of SC 514 (SIH-475), a IKK-2 kinase inhibitor. CAS #: 354812-17-2. Molecular Formula: C9H8N2OS2. Molecular Weight: 224.3 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of Nilotinib (SIH-463), a BCR-ABL kinase inhibitor. CAS #: 641571-10-0. Molecular Formula: C28H22F3N7O. Molecular Weight: 529.5 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of Auranofin (SIH-493), a IKK kinase inhibitor. CAS #: 34031-32-8. Molecular Formula: C20H34AuO9PS. Molecular Weight: 678.5 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
$87.00
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Chemical structure of ZM 336372 (SIH-488), a c-Raf kinase inhibitor. CAS #: 208260-29-1. Molecular Formula: C23H23N3O3. Molecular Weight: 389.4 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of Sorafenib (SIH-476), a Raf-1 inhibitor (and other kinases). CAS #: 2884461-73-0. Molecular Formula: C21H16ClF3N4O3. Molecular Weight: 464.8 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of WHI P131 (SIH-485), a JAK3 kinase inhibitor. CAS #: 202475-60-3. Molecular Formula: C16H15N3O3. Molecular Weight: 297.3 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of AR A014418 (SIH-492), a GSK-3 kinase inhibitor. CAS #: 487021-52-3. Molecular Formula: C12H12N4O4S. Molecular Weight: 308.3 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of Lestaurtinib (SIH-460), a FLT3/ TrkA kinase inhibitor. CAS #: 111358-88-4. Molecular Formula: C26H21N3O4. Molecular Weight: 439.5 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of BAY 11 7082 (SIH-434), a IKK kinase inhibitor. CAS #: 19542-67-7. Molecular Formula: C10H9NO2S. Molecular Weight: 207.3 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of A83 01 (SIH-423), a ALK kinase inhibitor. CAS #: 909910-43-6. Molecular Formula: C25H19N5S. Molecular Weight: 421.5 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of Genistein (SIH-446), a Tyrosine kinase inhibitor. CAS #: 446-72-0. Molecular Formula: C15H10O5. Molecular Weight: 270.2 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of AG 1517 (SIH-427), a EGFR tyrosine kinase inhibitor. CAS #: 153436-54-5. Molecular Formula: C16H14BrN3O2. Molecular Weight: 360.2 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of Flupirtine maleate (SIH-376), a Kv7 channel activator. CAS #: 75507-68-5. Molecular Formula: C15H17FN4O2.C4H4O4. Molecular Weight: 420.4 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $111.00
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Chemical structure of AS 041164 (SIH-433), a PI 3-Kgamma kinase inhibitor. CAS #: 6318-41-8. Molecular Formula: C11H7NO4S. Molecular Weight: 249.2 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of U-0126 (SIH-380), a MEK inhibitor. CAS #: 109511-58-2. Molecular Formula: C18H16N6S2. Molecular Weight: 380.5 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $170.00
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Chemical structure of Thiolutin (SIH-375), a HSP27 perturbing agent. CAS #: 87-11-6. Molecular Formula: C8H8N2O2S2. Molecular Weight: 228.3 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of Deprenyl (SIH-209), a glyceraldehyde-3-phosphate dehydrogenase inhibitor. CAS #: 14611-52-0. Molecular Formula: C13H17N · HCl . Molecular Weight: 223.74 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of Cycloheximide (SIH-247), a Translation inhibitor. CAS #: 66-81-9. Molecular Formula: C15H23NO4. Molecular Weight: 281.35 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
From $63.00
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