Cancer Biomarkers — Biochemicals

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Chemical structure of BSI 201 (SIH-539), a PARP1 inhibitor. CAS #: 160003-66-7. Molecular Formula: C7H5IN2O3. Molecular Weight: 292 g/mol.
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Chemical structure of LH 846 (SIH-503), a Casein kinase 1d inhibitor. CAS #: 639052-78-1. Molecular Formula: C16H13ClN2OS. Molecular Weight: 316.8 g/mol.
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Chemical structure of Ruxolitinib (SIH-509), a JAK kinase inhibitor. CAS #: 941678-49-5. Molecular Formula: C17H18N6. Molecular Weight: 306.4 g/mol.
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Chemical structure of Dovitinib (SIH-500), a FGFR3 inhibitor. CAS #: 405169-16-6. Molecular Formula: C21H21FN6O. Molecular Weight: 392.4 g/mol.
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Chemical structure of C8 Ceramide (SIH-499), a Protein kinase activator. CAS #: 74713-59-0. Molecular Formula: C26H51NO3. Molecular Weight: 425.7 g/mol.
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Chemical structure of BRD 7389 (SIH-497), a p90 RSK kinase inhibitor. CAS #: 376382-11-5. Molecular Formula: C24H18N2O2. Molecular Weight: 366.4 g/mol.
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Chemical structure of ZM 336372 (SIH-488), a c-Raf kinase inhibitor. CAS #: 208260-29-1. Molecular Formula: C23H23N3O3. Molecular Weight: 389.4 g/mol.
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Chemical structure of JX 401 (SIH-454), a p38alpha MAP kinase inhibitor. CAS #: 349087-34-9. Molecular Formula: C21H25NO2S. Molecular Weight: 355.5 g/mol.
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Chemical structure of K252A (SIH-455), a Kinase inhibitor (pan-specific). CAS #: 99533-80-9. Molecular Formula: C27H21N3O5. Molecular Weight: 467.5 g/mol.
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Chemical structure of GSK690693 Hydrochloride (SIH-448), a AKT kinase inhibitor. CAS #: 937174-76-0. Molecular Formula: C21H27N7O3. Molecular Weight: 425.5 g/mol.
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Chemical structure of A83 01 (SIH-423), a ALK kinase inhibitor. CAS #: 909910-43-6. Molecular Formula: C25H19N5S. Molecular Weight: 421.5 g/mol.
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Chemical structure of BzATP (SIH-420), a Prototypic P2X7 receptor agonist. CAS #: 112898-15-4. Molecular Formula: C24H24N5O15P3.C18H45N3. Molecular Weight: 1018.97 g/mol.
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Chemical structure of PHA 665752 (SIH-421), a MET kinase inhibitor. CAS #: 477575-56-7. Molecular Formula: C32H34Cl2N4O4S. Molecular Weight: 641.61 g/mol.
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Chemical structure of Deprenyl (SIH-209), a glyceraldehyde-3-phosphate dehydrogenase inhibitor. CAS #: 14611-52-0. Molecular Formula: C13H17N · HCl . Molecular Weight: 223.74 g/mol.
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Chemical structure of Mifepristone (RU486) (SIH-211), a Glucocorticoid antagonist. CAS #: 84371-65-3. Molecular Formula: C29H35NO2 . Molecular Weight: 429.6 g/mol.
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Chemical structure of Amifostine (SIH-210), a Cellular protectant. CAS #: 20537-88-6. Molecular Formula: C5H15N2O3PS. Molecular Weight: 214.22 g/mol.
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Chemical structure of bis-BHT (SIH-154), a Phenolic antioxidant. CAS #: 118-82-1. Molecular Formula: C29H44O2. Molecular Weight: 424.7 g/mol.
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Chemical structure of Deguelin (SIH-251), a Akt inhibitor. CAS #: 522-17-8. Molecular Formula: C23H22O6. Molecular Weight: 394.42 g/mol.
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Chemical structure of CCT241161 (SIH-186), a RAF Inhibitor. CAS #: 1163719-91-2. Molecular Formula: C28H27N7O3S. Molecular Weight: 541.63 g/mol.
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Chemical structure of Difluoromethylornithine (SIH-200), a Inhibits polyamine biosynthesis. CAS #: 70052-12-9. Molecular Formula: C6H12F2N2O2 * HCl. Molecular Weight: 218.63 g/mol.
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Chemical structure of 17-DMAG (SIH-114), a Hsp90 inhibitor. CAS #: 467214-20-6. Molecular Formula: C32H48N4O8. Molecular Weight: 616.8 g/mol.
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Chemical structure of Actinomycin D (SIH-245), a Transcription inhibitor. CAS #: 50-76-0. Molecular Formula: C62H86N12O16. Molecular Weight: 1255.43 g/mol.
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Chemical structure of 17-AAG (SIH-100), a Hsp90 inhibitor. CAS #: 75747-14-7. Molecular Formula: C31H43N3O8. Molecular Weight: 585.7 g/mol.
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Chemical structure of Felodipine (SIH-323), a L-type Ca channel blocker. CAS #: 72509-76-3. Molecular Formula: C18H19Cl2NO4. Molecular Weight: 384.25 g/mol.
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Chemical structure of TEMPO (SIH-155), a Stabilized free radical. CAS #: 2564-83-2. Molecular Formula: C9H18NO . Molecular Weight: 156.25 g/mol.
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Chemical structure of Geldanamycin- FITC (SIH-113), a Hsp90 inhibitor. Molecular Formula: C55H63N5O13S. Molecular Weight: 560.6 g/mol.
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Chemical structure of 17-GMB-APA-GA (SIH-115), a Hsp90 inhibitor. CAS #: N/A. Molecular Formula: C39H53N5O11. Molecular Weight: 767.9 g/mol.
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Chemical structure of Geldanamycin (SIH-111), a Hsp90 inhibitor. CAS #: 30562-34-6. Molecular Formula: C29H40N2O9. Molecular Weight: 560.6 g/mol.
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