Heat Shock Proteins & Chaperones

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1075 products
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Chemical structure of Dovitinib (SIH-500), a FGFR3 inhibitor. CAS #: 405169-16-6. Molecular Formula: C21H21FN6O. Molecular Weight: 392.4 g/mol.
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Chemical structure of C8 Ceramide (SIH-499), a Protein kinase activator. CAS #: 74713-59-0. Molecular Formula: C26H51NO3. Molecular Weight: 425.7 g/mol.
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Chemical structure of GW 441756 (SIH-450), a NGFR kinase inhibitor. CAS #: 504433-23-2. Molecular Formula: C17H13N3O. Molecular Weight: 275.3 g/mol.
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Chemical structure of JX 401 (SIH-454), a p38alpha MAP kinase inhibitor. CAS #: 349087-34-9. Molecular Formula: C21H25NO2S. Molecular Weight: 355.5 g/mol.
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Chemical structure of K252A (SIH-455), a Kinase inhibitor (pan-specific). CAS #: 99533-80-9. Molecular Formula: C27H21N3O5. Molecular Weight: 467.5 g/mol.
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Chemical structure of Quisqualic Acid (SIH-418), a Glutamate receptor agonist. CAS #: 52809-07-1. Molecular Formula: C5H7N3O5. Molecular Weight: 189.13 g/mol.
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Chemical structure of K252B (SIH-456), a Kinase inhibitor (pan-specific). CAS #: 99570-78-2. Molecular Formula: C26H19N3O5. Molecular Weight: 453.5 g/mol.
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Chemical structure of Dasatinib (SIH-440), a Src and Bcr/Abl kinase inhibitor. CAS #: 302962-49-8. Molecular Formula: C22H26ClN7O2S. Molecular Weight: 488 g/mol.
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Chemical structure of KT5720 (SIH-457), a PKA kinase inhibitor. CAS #: 108068-98-0. Molecular Formula: C32H31N3O5. Molecular Weight: 537.6 g/mol.
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Chemical structure of H89 Dihydrochloride (SIH-452), a PKA inhibitor. CAS #: 127243-85-0. Molecular Formula: C20H22BrCl2N3O2S. Molecular Weight: 519.3 g/mol.
H89
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Chemical structure of CID 2011756 (SIH-438), a PKD kinase inhibitor. CAS #: 638156-11-3. Molecular Formula: C22H21ClN2O3. Molecular Weight: 396.9 g/mol.
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Chemical structure of GSK690693 Hydrochloride (SIH-448), a AKT kinase inhibitor. CAS #: 937174-76-0. Molecular Formula: C21H27N7O3. Molecular Weight: 425.5 g/mol.
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Chemical structure of Imatinib mesylate (SIH-453), a BCR-ABL kinase inhibitor. CAS #: 152459-95-5. Molecular Formula: C30H35N7O4S. Molecular Weight: 589.7 g/mol.
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Chemical structure of GW2580 (SIH-449), a cFMS kinase inhibitor. CAS #: 870483-87-7. Molecular Formula: C20H22N4O3. Molecular Weight: 366.4 g/mol.
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Chemical structure of A83 01 (SIH-423), a ALK kinase inhibitor. CAS #: 909910-43-6. Molecular Formula: C25H19N5S. Molecular Weight: 421.5 g/mol.
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Chemical structure of Flupirtine maleate (SIH-376), a Kv7 channel activator. CAS #: 75507-68-5. Molecular Formula: C15H17FN4O2.C4H4O4. Molecular Weight: 420.4 g/mol.
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Chemical structure of BzATP (SIH-420), a Prototypic P2X7 receptor agonist. CAS #: 112898-15-4. Molecular Formula: C24H24N5O15P3.C18H45N3. Molecular Weight: 1018.97 g/mol.
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Chemical structure of PHA 665752 (SIH-421), a MET kinase inhibitor. CAS #: 477575-56-7. Molecular Formula: C32H34Cl2N4O4S. Molecular Weight: 641.61 g/mol.
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Chemical structure of 6BIO (SIH-422), a ESC self-renewal. CAS #: 667463-62-9. Molecular Formula: C16H10BrN3O2. Molecular Weight: 356.2 g/mol.
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Chemical structure of AAL 993 (SIH-424), a VEGFR inhibitor. CAS #: N/A. Molecular Formula: C20H16F3N3O. Molecular Weight: 371.4 g/mol.
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Chemical structure of Thiolutin (SIH-375), a HSP27 perturbing agent. CAS #: 87-11-6. Molecular Formula: C8H8N2O2S2. Molecular Weight: 228.3 g/mol.
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Chemical structure of IOX1 (SIH-377), a JMJD inhibitor. CAS #: 5852-78-8. Molecular Formula: C10H7 NO3. Molecular Weight: 189.2 g/mol.
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Chemical structure of Deprenyl (SIH-209), a glyceraldehyde-3-phosphate dehydrogenase inhibitor. CAS #: 14611-52-0. Molecular Formula: C13H17N · HCl . Molecular Weight: 223.74 g/mol.
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Chemical structure of Mifepristone (RU486) (SIH-211), a Glucocorticoid antagonist. CAS #: 84371-65-3. Molecular Formula: C29H35NO2 . Molecular Weight: 429.6 g/mol.
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Chemical structure of Piperlongumine (SIH-156), a Apoptosis inducer in oxidative stressed cells. CAS #: 20069-09-4. Molecular Formula: C17H19NO5. Molecular Weight: 317.3 g/mol.
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Chemical structure of Rapamycin (SIH-212), a mTOR inhibitor. CAS #: 53123-88-9. Molecular Formula: C51H79NO13 . Molecular Weight: 914.18 g/mol.
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Chemical structure of Amifostine (SIH-210), a Cellular protectant. CAS #: 20537-88-6. Molecular Formula: C5H15N2O3PS. Molecular Weight: 214.22 g/mol.
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Chemical structure of Mitomycin C (SIH-246), a DNA crosslinking and damaging agent. CAS #: 50-07-7. Molecular Formula: C15H18N4O5. Molecular Weight: 334.33 g/mol.
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Chemical structure of TPEN (SIH-231), a Intracellular Zn2+ chelator. CAS #: 16858-02-9. Molecular Formula: C26H28N6. Molecular Weight: 424.6 g/mol.
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Chemical structure of N,N-Dimethylsphingosine (SIH-235), a Inhibits sphingosine kinase. CAS #: 119567-63-4. Molecular Formula: C20H41NO2. Molecular Weight: 327.6 g/mol.
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Chemical structure of bis-BHT (SIH-154), a Phenolic antioxidant. CAS #: 118-82-1. Molecular Formula: C29H44O2. Molecular Weight: 424.7 g/mol.
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Chemical structure of Deguelin (SIH-251), a Akt inhibitor. CAS #: 522-17-8. Molecular Formula: C23H22O6. Molecular Weight: 394.42 g/mol.
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Chemical structure of CCT241161 (SIH-186), a RAF Inhibitor. CAS #: 1163719-91-2. Molecular Formula: C28H27N7O3S. Molecular Weight: 541.63 g/mol.
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Chemical structure of Camptothecin (SIH-242), a Topoisomerase I inhibitor. CAS #: 7689-03-4. Molecular Formula: C20H16N2O4. Molecular Weight: 348.36 g/mol.
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Chemical structure of Radicicol (SIH-117), a Hsp90 inhibitor. CAS #: 12772-57-5. Molecular Formula: C18H17CIO6. Molecular Weight: 364.8 g/mol.
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Chemical structure of Difluoromethylornithine (SIH-200), a Inhibits polyamine biosynthesis. CAS #: 70052-12-9. Molecular Formula: C6H12F2N2O2 * HCl. Molecular Weight: 218.63 g/mol.
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About Heat Shock Proteins & Chaperones

Antibodies, ELISA kits, and recombinant proteins for studying molecular chaperones, the heat shock response, and protein quality control. The category covers the major chaperone families — HSP90 (HSP90AA1, HSP90AB1, GRP94/HSP90B1, TRAP1/HSP75), HSP70 (HSPA1A, HSPA8, HSPA9/mortalin, GRP78/HSPA5), the small heat shock proteins (HSP27/HSPB1 and HSPB2–HSPB8), the chaperonins (HSP60/HSPD1 and HSP10), and the DNAJ/HSP40 co-chaperones — together with the HSP90 co-chaperone machinery (CDC37, HOP/STIP1, p23/PTGES3, AHA1/AHSA1) and the transcription factor HSF1 that drives the heat shock response. Use it to source validated reagents for proteostasis, chaperone-inhibitor, and cellular-stress research across human and preclinical species.

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