StressMarq Biosciences

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Chemical structure of Indirubin-3'-monoxime (SIH-502), a GSK-3b and CDK kinase inhibitor. CAS #: 160807-49-8. Molecular Formula: C16H11N3O2. Molecular Weight: 277.3 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of SU 4312 (SIH-481), a VEGFR / PDGFR kinase inhibitor. CAS #: 5812-07-7. Molecular Formula: C17H16N2O. Molecular Weight: 264.3 g/mol.
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Chemical structure of SR 3576 (SIH-513), a JNK3 kinase inhibitor. CAS #: 1164153-22-3. Molecular Formula: C27H27N5O5. Molecular Weight: 501.5 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of Dovitinib (SIH-500), a FGFR3 inhibitor. CAS #: 405169-16-6. Molecular Formula: C21H21FN6O. Molecular Weight: 392.4 g/mol.
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Chemical structure of PMA (SIH-508), a PKC kinase activator. CAS #: 16561-29-8. Molecular Formula: C36H58O8. Molecular Weight: 616.8 g/mol.
PMA
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of STO 609 (SIH-479), a CAMKK kinase inhibitor. CAS #: 52029-86-4. Molecular Formula: C21H14N2O5. Molecular Weight: 374.3 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of KT 5823 (SIH-458), a PKG kinase inhibitor. CAS #: 126643-37-6. Molecular Formula: C29H25N3O5. Molecular Weight: 495.5 g/mol.
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Chemical structure of AG 494 (SIH-491), a EGF receptor tyrosine kinase inhibitor. CAS #: 133550-35-3. Molecular Formula: C16H12N2O3. Molecular Weight: 280.3 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of SC 514 (SIH-475), a IKK-2 kinase inhibitor. CAS #: 354812-17-2. Molecular Formula: C9H8N2OS2. Molecular Weight: 224.3 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of C8 Ceramide (SIH-499), a Protein kinase activator. CAS #: 74713-59-0. Molecular Formula: C26H51NO3. Molecular Weight: 425.7 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of BIBW 2992 (SIH-496), a EGFR and HER2 kinase inhibitor. CAS #: 439081-18-2. Molecular Formula: C24H25ClFN5O3. Molecular Weight: 485.9 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of C16 (SIH-498), a PKR kinase inhibitor. CAS #: 608512-97-6. Molecular Formula: C13H8N4OS. Molecular Weight: 268.3 g/mol.
C16
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of Sunitinib malate (SIH-482), a VEGFR, PDGFR kinase inhibitor. CAS #: 557795-19-4. Molecular Formula: C22H27FN4O2. Molecular Weight: 398.5 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of Axitinib (SIH-494), a VEGFR kinase inhibitor. CAS #: 319460-85-0. Molecular Formula: C22H18N4OS. Molecular Weight: 386.5 g/mol.
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Chemical structure of SB203580 (SIH-474), a p38 MAP kinase inhibitor. CAS #: 152121-47-6. Molecular Formula: C21H16FN3OS. Molecular Weight: 377.4 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of Nilotinib (SIH-463), a BCR-ABL kinase inhibitor. CAS #: 641571-10-0. Molecular Formula: C28H22F3N7O. Molecular Weight: 529.5 g/mol.
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Chemical structure of BRD 7389 (SIH-497), a p90 RSK kinase inhibitor. CAS #: 376382-11-5. Molecular Formula: C24H18N2O2. Molecular Weight: 366.4 g/mol.
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Chemical structure of A 769662 (SIH-490), a AMPK kinase activator. CAS #: 844499-71-4. Molecular Formula: C20H12N2O3S. Molecular Weight: 360.4 g/mol.
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Chemical structure of Auranofin (SIH-493), a IKK kinase inhibitor. CAS #: 34031-32-8. Molecular Formula: C20H34AuO9PS. Molecular Weight: 678.5 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of ZM 336372 (SIH-488), a c-Raf kinase inhibitor. CAS #: 208260-29-1. Molecular Formula: C23H23N3O3. Molecular Weight: 389.4 g/mol.
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Chemical structure of GW 441756 (SIH-450), a NGFR kinase inhibitor. CAS #: 504433-23-2. Molecular Formula: C17H13N3O. Molecular Weight: 275.3 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of BML 259 (SIH-435), a CDK5/p25 kinase inhibitor. CAS #: 267654-00-2. Molecular Formula: C14H16N2OS. Molecular Weight: 260.4 g/mol.
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Chemical structure of JX 401 (SIH-454), a p38alpha MAP kinase inhibitor. CAS #: 349087-34-9. Molecular Formula: C21H25NO2S. Molecular Weight: 355.5 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of PX 866 (SIH-471), a PI 3-Kinase inhibitor. CAS #: 502632-66-8. Molecular Formula: C29H35NO8. Molecular Weight: 525.6 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of Erlotinib Hydrochloride (SIH-444), a EGFR Kinase inhibitor. CAS #: 183319-69-9. Molecular Formula: C22H24ClN3O4. Molecular Weight: 429.9 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of K252A (SIH-455), a Kinase inhibitor (pan-specific). CAS #: 99533-80-9. Molecular Formula: C27H21N3O5. Molecular Weight: 467.5 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of Src I1 (SIH-478), a Src kinase inhibitor. CAS #: 179248-59-0. Molecular Formula: C22H19N3O3. Molecular Weight: 373.4 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of Sorafenib (SIH-476), a Raf-1 inhibitor (and other kinases). CAS #: 2884461-73-0. Molecular Formula: C21H16ClF3N4O3. Molecular Weight: 464.8 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of Quisqualic Acid (SIH-418), a Glutamate receptor agonist. CAS #: 52809-07-1. Molecular Formula: C5H7N3O5. Molecular Weight: 189.13 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of WHI P131 (SIH-485), a JAK3 kinase inhibitor. CAS #: 202475-60-3. Molecular Formula: C16H15N3O3. Molecular Weight: 297.3 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of AR A014418 (SIH-492), a GSK-3 kinase inhibitor. CAS #: 487021-52-3. Molecular Formula: C12H12N4O4S. Molecular Weight: 308.3 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of LFM A13 (SIH-461), a BTK kinase inhibitor. CAS #: 62004-35-7. Molecular Formula: C11H8Br2N2O2. Molecular Weight: 360 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of ZM447439 (SIH-489), a Aurora B kinase inhibitor. CAS #: 331771-20-1. Molecular Formula: C29H31N5O4. Molecular Weight: 513.6 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of NPC 15437 (SIH-464), a PKC kinase inhibitor. CAS #: 141774-20-1. Molecular Formula: C25H52Cl2N4O2. Molecular Weight: 511.6 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of Midostaurin (SIH-468), a Protein kinase inhibitor (pan spec.). CAS #: 120685-11-2. Molecular Formula: C35H30N4O4. Molecular Weight: 570.6 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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Chemical structure of GW5074 (SIH-451), a c-Raf1 kinase inhibitor. CAS #: 220904-83-6. Molecular Formula: C15H8Br2INO2. Molecular Weight: 520.9 g/mol.
Biochemicals, Small Molecules Functional Assay (In Vitro)
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